含氮杂环化合物的合成和结构具有极大吸引力，因为这些化合物结构丰富、理化性质和生物性质多样。因此，开发改进方法，合成多官能团含氮杂环化合物一直是一个具有挑战性的目标。本文描述了在过去 15 年中，我们的实验室在发现 C-H/N-H 键官能化和含氮杂环化合物（氮丙啶类、吲哚类、中氮茚类、三唑类、咪唑类、噁唑、噻唑类、喹喔啉、三嗪类和吡啶类）合成中的氧化环化途径中的探索。

The synthesis and structure of nitrogen-containing heterocycles are fascinating because these compounds have a great richness of structural, physicochemical, and biological properties. Therefore, the development of improved ways for the synthesis of polyfunctional nitrogen-containing heterocycles continues to be a challenging goal. This account describes developments in the discovery of C–H/N–H bond functionalization and oxidative cyclization procedures for the synthesis of nitrogen-containing heterocycles (aziridines, indoles, indolizines, triazoles, imidazoles, oxazoles, thiazoles, quinoxalines, triazines, and pyridines) in our laboratories during the last 15 years.